{"id":416426,"date":"2026-03-10T18:00:00","date_gmt":"2026-03-10T10:00:00","guid":{"rendered":"https:\/\/pingtungtimes.com.tw\/?p=416426"},"modified":"2026-03-10T18:00:00","modified_gmt":"2026-03-10T10:00:00","slug":"%e6%ad%8c%e7%a6%ae%e5%ae%a3%e4%bd%88%e5%85%b6%e5%b0%8f%e5%88%86%e5%ad%90glp-1r%e6%bf%80%e5%8b%95%e5%8a%91asc30%e7%9a%84%e8%b6%85%e9%95%b7%e6%95%88%e7%9a%ae%e4%b8%8b%e5%84%b2%e5%ba%ab%e5%9e%8b%e5%88%b6","status":"publish","type":"post","link":"https:\/\/pingtungtimes.com.tw\/?p=416426","title":{"rendered":"\u6b4c\u79ae\u5ba3\u4f48\u5176\u5c0f\u5206\u5b50GLP-1R\u6fc0\u52d5\u5291ASC30\u7684\u8d85\u9577\u6548\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u91dd\u5c0d\u80a5\u80d6\u9069\u61c9\u75c7\u7684\u7f8e\u570bII\u671f24\u5468\u7814\u7a76\u7372\u7a4d\u6975\u9802\u7dda\u7d50\u679c"},"content":{"rendered":"<div>\n<p><i>&#8211; \u00a0 \u00a0ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u5728\u6bcf\u67081\u6b21\u3001\u5171\u8a083\u6b21\u7d66\u85e5\u5f8c\uff0c\u5728\u7b2c16\u5468\u5be6\u73fe\u4e86\u5177\u6709\u7d71\u8a08\u5b78\u986f\u8457\u6027\u548c\u81e8\u5e8a\u610f\u7fa9\u7684\u5e73\u5747\u9ad4\u91cd\u4e0b\u964d7.5%\uff08\u7d93\u5b89\u6170\u5291\u6821\u6b63\u5f8c\uff09\u3002<\/p>\n<p>&#8211; \u00a0 \u00a0ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u7b2c\u4e09\u6b21\u5373\u672b\u6b21\u6bcf\u6708\u4e00\u6b21\u7d66\u85e5\u5f8c\uff0c\u6e1b\u91cd\u6548\u679c\u7dad\u6301\u9577\u90544\u500b\u6708\uff0c\u8868\u660e\u5176\u6709\u671b\u4f5c\u70ba\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7d66\u85e5\u7684\u7dad\u6301\u7642\u6cd5\u3002<\/p>\n<p>&#8211; \u00a0 \u00a0ASC30\u986f\u793a\u51fa\u7684\u5b89\u5168\u6027\u548c\u8010\u53d7\u6027\u7279\u5fb5\u8207GLP-1\u985e\u85e5\u7269\u7684\u4e00\u81f4\u3002<\/p>\n<p>&#8211; \u00a0 \u00a0ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u662f\u9996\u6b3e\u7121\u9700\u6bcf\u9031\u4e00\u6b21\u6ce8\u5c04\u7684\u6e96\u5099\uff08lead-in\uff09\u671f\u3001\u76f4\u63a5\u6bcf\u6708\u4e00\u6b21\u6ce8\u5c04\u5373\u53ef\u5be6\u73fe\u8207\u540c\u985e\u85e5\u7269\u4e00\u81f4\u7684\u6e1b\u91cd\u6548\u679c\uff0c\u4e14\u672b\u6b21\u7d66\u85e5\u5f8c\u6e1b\u91cd\u6548\u679c\u53ef\u7dad\u6301\u9577\u90544\u500b\u6708\u7684GLP-1\u85e5\u7269\u3002<\/i><\/p>\n<p><span class=\"legendSpanClass\">\u9999\u6e2f<\/span><span class=\"legendSpanClass\">2026\u5e743\u670810\u65e5<\/span> \/\u7f8e\u901a\u793e\/ &#8212; \u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8\uff08\u9999\u6e2f\u806f\u4ea4\u6240\u4ee3\u78bc\uff1a1672\uff0c\u7c21\u7a31\u300c\u6b4c\u79ae\u300d\uff09\u5ba3\u4f48\uff0c\u5176\u5c0f\u5206\u5b50GLP-1\u53d7\u9ad4\uff08GLP-1R\uff09\u6fc0\u52d5\u5291ASC30\u76ae\u4e0b\u5132\u5eab\u578b\uff08depot\uff09\u5236\u5291\u91dd\u5c0d\u80a5\u80d6\u9069\u61c9\u75c7\u7684\u7f8e\u570bII\u671f24\u5468\u7814\u7a76\uff08<a href=\"https:\/\/clinicaltrials.gov\/study\/NCT06679959?cond=ASC30&amp;rank=3\" target=\"_blank\" rel=\"nofollow\" style=\"color: #0000FF\">NCT06679959<\/a>\uff09\u53d6\u5f97\u7a4d\u6975\u9802\u7dda\u7d50\u679c\u3002\u4e09\u500b\u968a\u5217\u5171\u5165\u7d4465\u540d\u53d7\u8a66\u8005\uff0c\u63a1\u7528\u5169\u7a2e\u5236\u5291\uff08A1\u548cA2\uff09\u7d66\u85e5\uff0c\u6240\u6709\u53d7\u8a66\u8005\u5747\u70ba\u80a5\u80d6\u53d7\u8a66\u8005\u6216\u4f34\u6709\u81f3\u5c11\u4e00\u7a2e\u9ad4\u91cd\u76f8\u95dc\u5408\u4f75\u75c7\u7684\u8d85\u91cd\u53d7\u8a66\u8005\u3002<\/p>\n<p>\u8a72II\u671f\u7814\u7a76\u9054\u5230\u4e86\u5176\u4e3b\u8981\u7d42\u9ede\uff0c\u63a5\u53d73\u5291\uff08\u6bcf\u6708\u4e00\u6b21\uff09ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u7684\u60a3\u8005<span id=\"spanHghlt2176\">\u5728<\/span>\u7b2c12\u5468\u986f\u793a\u51fa\u5177\u6709\u7d71\u8a08\u5b78\u986f\u8457\u6027\uff08\u5c0d\u6bd4\u5b89\u6170\u5291\uff0c<i>p<\/i>&lt;0.05\uff09\u548c\u81e8\u5e8a\u610f\u7fa9\u7684\u5e73\u5747\u9ad4\u91cd\u4e0b\u964d6.3%\uff08\u7d93\u5b89\u6170\u5291\u6821\u6b63\u5f8c\uff09\u3002\u6b64\u5916\uff0cASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u5728\u6bcf\u67081\u6b21\u3001\u5171\u8a083\u6b21\u7d66\u85e5\u5f8c\uff0c\u5728\u7b2c16\u5468\u986f\u793a\u51fa\u5177\u6709\u7d71\u8a08\u5b78\u986f\u8457\u6027\uff08\u5c0d\u6bd4\u5b89\u6170\u5291\uff0c<i>p<\/i>&lt;0.05\uff09\u548c\u81e8\u5e8a\u610f\u7fa9\u7684\u5e73\u5747\u9ad4\u91cd\u4e0b\u964d7.5%\uff08\u7d93\u5b89\u6170\u5291\u6821\u6b63\u5f8c\uff09\u3002<\/p>\n<p>\u8a72II\u671f\u7814\u7a76\u70ba\u4e00\u9805\u5728\u7f8e\u570b\u958b\u5c55\u7684\u96a8\u6a5f\u3001\u96d9\u76f2\u3001\u5b89\u6170\u5291\u5c0d\u7167\u53ca\u591a\u4e2d\u5fc3\u7684\u70ba\u671f24\u5468\u7684\u7814\u7a76\uff0c\u65e8\u5728\u8a55\u4f30ASC30\u572865\u4f8b\u80a5\u80d6\u53d7\u8a66\u8005\uff08\u9ad4\u91cd\u6307\u6578BMI \u2265 30 kg\/m\u00b2\uff09\u6216\u4f34\u6709\u81f3\u5c11\u4e00\u7a2e\u9ad4\u91cd\u76f8\u95dc\u5408\u4f75\u75c7\u7684\u8d85\u91cd\u53d7\u8a66\u8005\uff0827 kg\/m\u00b2 \u2264 BMI &lt; 30 kg\/m\u00b2\uff09\u4e2d\u7684\u5b89\u5168\u6027\u3001\u8010\u53d7\u6027\u53ca\u7642\u6548\u300265\u4f8b\u53d7\u8a66\u8005\u5747\u5728\u7b2c1\u5929\u3001\u7b2c29\u5929\uff08\u7b2c4\u5468\uff09\u53ca\u7b2c57\u5929\uff08\u7b2c8\u5468\uff09\u63a5\u53d7\u6bcf\u6708\u4e00\u6b21\u7684ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u6216\u5339\u914d\u7684\u5b89\u6170\u5291\u7d66\u85e5\uff08\u51713\u5291\uff09\uff0c\u7121\u9700\u6bcf\u9031\u4e00\u6b21\u7d66\u85e5\u7684\u6e96\u5099\uff08lead-in\uff09\u671f\u3002\u7dad\u6301\u671f\u5f9e\u7b2c8\u5468\u958b\u59cb\u81f3\u7b2c24\u5468\uff0c\u517116\u5468\u3002\u8a72\u7814\u7a76\u5c0dASC30\u7684\u5169\u7a2e\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\uff08A1\u548cA2\uff09\u9032\u884c\u4e86\u8a55\u4f30\uff0c\u7814\u7a76\u76ee\u7684\u70ba\u8a55\u4f30\u6bcf\u6708\u4e00\u6b21\u7d66\u85e5\u7684\u6cbb\u7642\u7642\u6cd5\u548c\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7d66\u85e5\u7684\u7dad\u6301\u7642\u6cd5\u7684\u6f5b\u529b\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u6b64\u524d\u5df2\u5728\u4e00\u9805\u70ba\u671f12\u5468\u7684Ib\u671f\u55ae\u5291\u91cf\u7814\u7a76\uff08<a href=\"https:\/\/clinicaltrials.gov\/study\/NCT06679959?cond=ASC30&amp;rank=3\" target=\"_blank\" rel=\"nofollow\" style=\"color: #0000FF\">NCT06679959<\/a>\uff09\u4e2d\u9032\u884c\u8a55\u4f30\uff0c\u7d50\u679c\u986f\u793a\u5176\u8868\u89c0\u534a\u8870\u671f\uff08observed half-life\uff09\u70ba46\u5929\u81f375\u5929\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A2\u6b64\u524d\u5c1a\u672a\u958b\u5c55\u904e\u4eba\u9ad4\u7814\u7a76\u3002\u5728\u672c\u7814\u7a76\u4e2d\uff0c\u5236\u5291A1\u5728\u80a5\u80d6\u60a3\u8005\u4e2d\u9054\u5230\u4e86\u6cbb\u7642\u6027\u85e5\u7269\u66b4\u9732\u6c34\u5e73\uff08therapeutic drug exposures\uff09\uff0c\u800c\u5236\u5291A2\u672a\u9054\u5230\u3002<\/p>\n<p>ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u7684\u7d66\u85e5\u65b9\u6848\uff1a\u6240\u6709\u53d7\u8a66\u8005\u63a5\u53d7\u4e09\u6b21\u76ae\u4e0b\u7d66\u85e5\uff0c\u7d66\u85e5\u9593\u9694\u70ba\u56db\u5468\uff0c\u5206\u5225\u5728\u7b2c1\u5929\u3001\u7b2c29\u5929\uff08\u7b2c4\u5468\uff09\u548c\u7b2c57\u5929\uff08\u7b2c8\u5468\uff09\u7d66\u85e5\uff0c\u6bcf\u6b21\u5291\u91cf\u70ba400\u6beb\u514b\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u5728\u7b2c4\u5468\u3001\u7b2c8\u5468\u3001\u7b2c12\u5468\u548c\u7b2c16\u5468\u5206\u5225\u5be6\u73fe\u4e862.7%\u30015.5%\u30016.3%\u548c7.5%\u7684\u7d93\u5b89\u6170\u5291\u6821\u6b63\u5f8c\u7684\u5e73\u5747\u9ad4\u91cd\u4e0b\u964d\u3002\u9019\u4e9b\u6578\u64da\u986f\u793a\uff0cASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u53ef\u6bcf\u6708\u4e00\u6b21\u7d66\u85e5\u7528\u65bc\u80a5\u80d6\u75c7\u6cbb\u7642\uff0c\u4e26\u6709\u671b\u5be6\u73fe\u6bcf\u5169\u500b\u6708\u4e00\u6b21\u7d66\u85e5\uff0c\u4e14\u7121\u9700\u6bcf\u9031\u4e00\u6b21\u7d66\u85e5\u7684\u6e96\u5099\u671f\u3002<\/p>\n<p>\u8a72II\u671f\u7814\u7a76\u540c\u6642\u8a55\u4f30\u4e86ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u4f5c\u70ba\u7dad\u6301\u7642\u6cd5\u7684\u6f5b\u529b\u3002\u5728\u7b2c8\u5468\u5b8c\u6210\u672b\u6b21\u7d66\u85e5\u5f8c\uff0c\u5c0d\u5728\u60a3\u8005\u4e2d\u7684\u7642\u6548\u6301\u7e8c\u6642\u9593\u9032\u884c\u4e86\u70ba\u671f16\u5468\u7684\u8a55\u4f30\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u5728\u672b\u6b21\u7d66\u85e5\u5f8c\u768416\u5468\u7dad\u6301\u671f\u5167\u5747\u9054\u5230\u4e86\u6cbb\u7642\u6027\u85e5\u7269\u66b4\u9732\u6c34\u5e73\u3002\u7d93\u5b89\u6170\u5291\u6821\u6b63\u5f8c\u7684\u5e73\u5747\u9ad4\u91cd\u4e0b\u964d\u5728\u7b2c8\u5468\u70ba5.5%\uff0c\u7b2c20\u5468\uff08\u672b\u6b21\u7d66\u85e5\u5f8c3\u500b\u6708\uff09\u70ba6.4%\uff0c\u7b2c24\u5468\uff08\u672b\u6b21\u7d66\u85e5\u5f8c4\u500b\u6708\uff09\u70ba5.8%\u3002\u9019\u4e9b\u7d50\u679c\u986f\u793aASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u6709\u671b\u6210\u70ba\u6bcf\u5b63\u5ea6\u7d66\u85e5\u4e00\u6b21\u7684\u6709\u6548\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\u3002<\/p>\n<p>ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u548cA2\u5b89\u5168\u6027\u548c\u8010\u53d7\u6027\u826f\u597d\uff0c\u5176\u5b89\u5168\u6027\u548c\u8010\u53d7\u6027\u7279\u5fb5\u548cGLP\u20111\u985e\u85e5\u7269\u4e00\u81f4\u3002\u7d93ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u548cA2\u6216\u5b89\u6170\u5291\u6cbb\u7642\u7684\u53d7\u8a66\u8005\u5747\u7121\u56e0\u4e0d\u826f\u4e8b\u4ef6\uff08AE\uff09\u800c\u505c\u85e5\u7684\u60c5\u6cc1\u3002\u6240\u6709\u4e0d\u826f\u4e8b\u4ef6\uff08\u5305\u62ec\u6ce8\u5c04\u90e8\u4f4d\u4e0d\u826f\u4e8b\u4ef6\uff09\u7684\u56b4\u91cd\u7a0b\u5ea6\u5747\u70ba\u8f15\u5ea6\u81f3\u4e2d\u5ea6\u3002\u6240\u6709\u80c3\u8178\u9053\uff08GI\uff09\u4e0d\u826f\u4e8b\u4ef6\u5747\u70ba\u8f15\u5ea6\uff081\u7d1a\uff09\uff0c\u7121\u4e2d\u5ea6\uff082\u7d1a\uff09\u53ca\u4ee5\u4e0a\u80c3\u8178\u9053\u4e0d\u826f\u4e8b\u4ef6\u3002\u672a\u89c0\u5bdf\u5230\u809d\u81df\u5b89\u5168\u6027\u4fe1\u865f\u3002\u6b64\u5916\uff0c\u5be6\u9a57\u5ba4\u6aa2\u67e5\u3001\u751f\u547d\u9ad4\u5f81\u3001\u5fc3\u96fb\u5716\uff08\u5305\u62ecQTc\u9593\u671f\uff09\u548c\u9ad4\u683c\u6aa2\u67e5\u5747\u672a\u898b\u7570\u5e38\u7d50\u679c\u3002<\/p>\n<p>\u300c\u5728\u63a5\u53d7ASC30\u9577\u6548\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u6cbb\u7642\u7684\u80a5\u80d6\u60a3\u8005\u4e2d\u89c0\u5bdf\u5230\u5177\u6709\u7d71\u8a08\u5b78\u986f\u8457\u6027\u548c\u81e8\u5e8a\u610f\u7fa9\u7684\u9ad4\u91cd\u4e0b\u964d\uff0c\u6211\u5011\u6df1\u611f\u632f\u596e\u3002ASC30\u65e2\u53ef\u4f5c\u70ba\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u7d66\u85e5\u6216\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u7d66\u85e5\u7684\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\uff0c\u4e5f\u53ef\u4f5c\u70ba\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u7d66\u85e5\u7684\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u662f\u9996\u6b3e\u4e5f\u662f\u552f\u4e00\u4e00\u6b3e\u64c1\u6709\u4e0a\u8ff0\u7d66\u85e5\u983b\u7387\u548c\u7d66\u85e5\u9014\u5f91\u4e26\u5df2\u5728\u5169\u9805II\u671f\u7814\u7a76\u4e2d\u8b49\u660e\u53ef\u5be6\u73fe\u6709\u6548\u6e1b\u91cd\u7684\u8178\u4fc3\u80f0\u7d20\uff08incretin\uff09\u3002\u300d\u6b4c\u79ae\u5275\u59cb\u4eba\u3001\u8463\u4e8b\u6703\u4e3b\u5e2d\u517c\u9996\u5e2d\u57f7\u884c\u5b98\u5433\u52c1\u6893\u535a\u58eb\u8868\u793a\uff0c\u300cASC30\u9577\u6548\u5236\u5291\u517c\u5177\u5177\u6709\u7af6\u722d\u529b\u7684\u7642\u6548\u8207\u826f\u597d\u7684\u5b89\u5168\u6027\u3001\u8010\u53d7\u6027\u7279\u5fb5\uff0c\u9019\u9032\u4e00\u6b65\u589e\u5f37\u4e86\u6211\u5011\u64f4\u5927ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u81e8\u5e8a\u958b\u767c\u9805\u76ee\u7684\u4fe1\u5fc3\uff0c\u5305\u62ec\u6bcf\u6708\u4e00\u6b21\u7684\u6cbb\u7642\u7642\u6cd5\uff0c\u4ee5\u53ca\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7684\u7dad\u6301\u7642\u6cd5\u3002\u6b64\u5916\uff0c\u5f9e\u9019\u9805\u70ba\u671f24\u5468\u3001\u4f7f\u7528\u6b4c\u79ae\u5c08\u6709\u7684\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u7684\u7814\u7a76\u4e2d\u7372\u5f97\u7684\u6578\u64da\uff0c\u9a57\u8b49\u4e86\u6b4c\u79ae\u8d85\u9577\u6548\u85e5\u7269\u958b\u767c\u5e73\u53f0\uff08Ultra-Long-Acting Platform\uff0cULAP\uff09\u6280\u8853\u5728\u958b\u767c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u7684\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7642\u6cd5\u7684\u53ef\u884c\u6027\u3002\u300d<\/p>\n<p>\u7531\u6b4c\u79ae\u81ea\u4e3b\u7814\u767c\u7684ASC30\u662f\u9996\u6b3e\u4e5f\u662f\u552f\u4e00\u4e00\u6b3e\u6b63\u5728\u81e8\u5e8a\u7814\u7a76\u4e2d\u7684\u3001\u65e2\u53ef\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u4e5f\u53ef\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u7684\u5c0f\u5206\u5b50GLP-1R\u504f\u5411\u6fc0\u52d5\u5291\uff0c\u65e2\u53ef\u4f5c\u70ba\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\u4e5f\u53ef\u4f5c\u70ba\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u3002<\/p>\n<p><b>\u95dc\u65bc<\/b><b>ASC30<\/b><\/p>\n<p>ASC30\u662f\u4e00\u6b3e\u6b63\u5728\u81e8\u5e8a\u7814\u7a76\u4e2d\u7684\u5c0f\u5206\u5b50GLP-1R\u504f\u5411\u6fc0\u52d5\u5291\uff0c\u5177\u6709\u7368\u7279\u548c\u5dee\u7570\u5316\u6027\u8cea\uff0c\u4f7f\u5f97\u540c\u4e00\u5c0f\u5206\u5b50\u540c\u6642\u9069\u7528\u65bc\u53e3\u670d\u7247\u5291\u548c\u76ae\u4e0b\u6ce8\u5c04\u7d66\u85e5\u6210\u70ba\u53ef\u80fd\u3002ASC30\u662f\u4e00\u7a2e\u65b0\u5316\u5b78\u5be6\u9ad4\uff08NCE\uff09\uff0c\u64c1\u6709\u7f8e\u570b\u548c\u5168\u7403\u5316\u5408\u7269\u5c08\u5229\u4fdd\u8b77\uff0c\u5c08\u5229\u4fdd\u8b77\u671f\u81f32044\u5e74\uff08\u4e0d\u542b\u6f5b\u5728\u7684\u5c08\u5229\u5ef6\u671f\uff09\u3002<\/p>\n<p><b>\u95dc\u65bc\u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8<\/b><\/p>\n<p>\u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8\u662f\u4e00\u5bb6\u5168\u50f9\u503c\u93c8\u6574\u5408\u578b\u751f\u7269\u6280\u8853\u516c\u53f8\uff0c\u805a\u7126\u6709\u671b\u6210\u70ba\u6cbb\u7642\u4ee3\u8b1d\u75be\u75c5\u540c\u985e\u6700\u4f73\uff08best-in-class\uff09\u548c\u540c\u985e\u9996\u5275\uff08first-in-class\uff09\u85e5\u7269\u7684\u958b\u767c\u548c\u5546\u696d\u5316\u3002\u5229\u7528\u516c\u53f8\u5c08\u6709\u7684\u57fa\u65bc\u7d50\u69cb\u7684AI\u8f14\u52a9\u85e5\u7269\u767c\u73fe\uff08Artificial Intelligence-assisted Structure-Based Drug Discovery\uff0cAISBDD\uff09\u3001\u8d85\u9577\u6548\u85e5\u7269\u958b\u767c\u5e73\u53f0\uff08Ultra-Long-Acting Platform\uff0cULAP\uff09\u6280\u8853\u4ee5\u53ca\u53e3\u670d\u591a\u80bd\u905e\u9001\u589e\u5f37\u6280\u8853\uff08Peptide Oral Transport ENhancement Technology\uff0cPOTENT\uff09\uff0c\u6b4c\u79ae\u5df2\u81ea\u4e3b\u7814\u767c\u591a\u6b3e\u5c0f\u5206\u5b50\u548c\u591a\u80bd\u5019\u9078\u85e5\u7269\uff0c\u5305\u62ec\u5176\u6838\u5fc3\u9805\u76eeASC30\uff0c\u4e00\u6b3e\u5728\u7814\u5c0f\u5206\u5b50GLP-1R\u6fc0\u52d5\u5291\uff0c\u65e2\u53ef\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u4e5f\u53ef\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u4f5c\u70ba\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\u548c\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\uff1bASC36\uff0c\u4e00\u6b3e\u80f0\u6fb1\u7d20\u53d7\u9ad4\u6fc0\u52d5\u5291\u591a\u80bd\uff0cASC35\uff0c\u4e00\u6b3e\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04GLP-1R\/GIPR\u96d9\u9776\u9ede\u6fc0\u52d5\u5291\u591a\u80bd\uff0cASC37\uff0c\u4e00\u6b3eGLP-1R\/GIPR\/GCGR\u4e09\u9776\u9ede\u6fc0\u52d5\u5291\u591a\u80bd\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u3002\u6b4c\u79ae\u5df2\u5728\u9999\u6e2f\u806f\u4ea4\u6240\u4e0a\u5e02\uff081672.HK\uff09\u3002<\/p>\n<p>\u6b32\u77ad\u89e3\u66f4\u591a\u4fe1\u606f\uff0c\u656c\u8acb\u767b\u9304\u7db2\u7ad9\uff1a<a href=\"https:\/\/www.ascletis.com\/\" target=\"_blank\" rel=\"nofollow\" style=\"color: #0000FF\">www.ascletis.com<\/a>\u3002<\/p>\n<p>\u8a73\u60c5\u5782\u8a62\uff1a<\/p>\n<p>Peter Vozzo<br \/>ICR Healthcare<br \/>443-231-0505 (\u7f8e\u570b)<br \/><a href=\"mailto:Peter.vozzo@icrhealthcare.com\" rel=\"nofollow\" style=\"color: #0000FF\">Peter.vozzo@icrhealthcare.com<\/a><\/p>\n<p>\u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8PR\u548cIR\u5718\u968a<br \/>+86-181-0650-9129 (\u4e2d\u570b)<br \/><a href=\"mailto:pr@ascletis.com\" target=\"_blank\" rel=\"nofollow\" style=\"color: #0000FF\">pr@ascletis.com<\/a><br \/><a href=\"mailto:ir@ascletis.com\" target=\"_blank\" rel=\"nofollow\" style=\"color: #0000FF\">ir@ascletis.com<\/a>\u00a0<\/p>\n<\/div>\n","protected":false},"excerpt":{"rendered":"<p>&#8211; \u00a0 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ASC30\u662f\u4e00\u6b3e\u6b63\u5728\u81e8\u5e8a\u7814\u7a76\u4e2d\u7684\u5c0f\u5206\u5b50GLP-1R\u504f\u5411\u6fc0\u52d5\u5291\uff0c\u5177\u6709\u7368\u7279\u548c\u5dee\u7570\u5316\u6027\u8cea\uff0c\u4f7f\u5f97\u540c\u4e00\u5c0f\u5206\u5b50\u540c\u6642\u9069\u7528\u65bc\u53e3\u670d\u7247\u5291\u548c\u76ae\u4e0b\u6ce8\u5c04\u7d66\u85e5\u6210\u70ba\u53ef\u80fd\u3002ASC30\u662f\u4e00\u7a2e\u65b0\u5316\u5b78\u5be6\u9ad4\uff08NCE\uff09\uff0c\u64c1\u6709\u7f8e\u570b\u548c\u5168\u7403\u5316\u5408\u7269\u5c08\u5229\u4fdd\u8b77\uff0c\u5c08\u5229\u4fdd\u8b77\u671f\u81f32044\u5e74\uff08\u4e0d\u542b\u6f5b\u5728\u7684\u5c08\u5229\u5ef6\u671f\uff09\u3002 \u95dc\u65bc\u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8 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Technology\uff0cPOTENT\uff09\uff0c\u6b4c\u79ae\u5df2\u81ea\u4e3b\u7814\u767c\u591a\u6b3e\u5c0f\u5206\u5b50\u548c\u591a\u80bd\u5019\u9078\u85e5\u7269\uff0c\u5305\u62ec\u5176\u6838\u5fc3\u9805\u76eeASC30\uff0c\u4e00\u6b3e\u5728\u7814\u5c0f\u5206\u5b50GLP-1R\u6fc0\u52d5\u5291\uff0c\u65e2\u53ef\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u4e5f\u53ef\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u4f5c\u70ba\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\u548c\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\uff1bASC36\uff0c\u4e00\u6b3e\u80f0\u6fb1\u7d20\u53d7\u9ad4\u6fc0\u52d5\u5291\u591a\u80bd\uff0cASC35\uff0c\u4e00\u6b3e\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04GLP-1R\/GIPR\u96d9\u9776\u9ede\u6fc0\u52d5\u5291\u591a\u80bd\uff0cASC37\uff0c\u4e00\u6b3eGLP-1R\/GIPR\/GCGR\u4e09\u9776\u9ede\u6fc0\u52d5\u5291\u591a\u80bd\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u3002\u6b4c\u79ae\u5df2\u5728\u9999\u6e2f\u806f\u4ea4\u6240\u4e0a\u5e02\uff081672.HK\uff09\u3002 \u6b32\u77ad\u89e3\u66f4\u591a\u4fe1\u606f\uff0c\u656c\u8acb\u767b\u9304\u7db2\u7ad9\uff1awww.ascletis.com\u3002 \u8a73\u60c5\u5782\u8a62\uff1a Peter VozzoICR Healthcare443-231-0505 (\u7f8e\u570b)Peter.vozzo@icrhealthcare.com \u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8PR\u548cIR\u5718\u968a+86-181-0650-9129 (\u4e2d\u570b)pr@ascletis.comir@ascletis.com\u00a0\" \/>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/pingtungtimes.com.tw\/?p=416426\" \/>\n<meta property=\"og:locale\" content=\"zh_TW\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u6b4c\u79ae\u5ba3\u4f48\u5176\u5c0f\u5206\u5b50GLP-1R\u6fc0\u52d5\u5291ASC30\u7684\u8d85\u9577\u6548\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u91dd\u5c0d\u80a5\u80d6\u9069\u61c9\u75c7\u7684\u7f8e\u570bII\u671f24\u5468\u7814\u7a76\u7372\u7a4d\u6975\u9802\u7dda\u7d50\u679c - 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kg\/m\u00b2\uff09\u4e2d\u7684\u5b89\u5168\u6027\u3001\u8010\u53d7\u6027\u53ca\u7642\u6548\u300265\u4f8b\u53d7\u8a66\u8005\u5747\u5728\u7b2c1\u5929\u3001\u7b2c29\u5929\uff08\u7b2c4\u5468\uff09\u53ca\u7b2c57\u5929\uff08\u7b2c8\u5468\uff09\u63a5\u53d7\u6bcf\u6708\u4e00\u6b21\u7684ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u6216\u5339\u914d\u7684\u5b89\u6170\u5291\u7d66\u85e5\uff08\u51713\u5291\uff09\uff0c\u7121\u9700\u6bcf\u9031\u4e00\u6b21\u7d66\u85e5\u7684\u6e96\u5099\uff08lead-in\uff09\u671f\u3002\u7dad\u6301\u671f\u5f9e\u7b2c8\u5468\u958b\u59cb\u81f3\u7b2c24\u5468\uff0c\u517116\u5468\u3002\u8a72\u7814\u7a76\u5c0dASC30\u7684\u5169\u7a2e\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\uff08A1\u548cA2\uff09\u9032\u884c\u4e86\u8a55\u4f30\uff0c\u7814\u7a76\u76ee\u7684\u70ba\u8a55\u4f30\u6bcf\u6708\u4e00\u6b21\u7d66\u85e5\u7684\u6cbb\u7642\u7642\u6cd5\u548c\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7d66\u85e5\u7684\u7dad\u6301\u7642\u6cd5\u7684\u6f5b\u529b\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u6b64\u524d\u5df2\u5728\u4e00\u9805\u70ba\u671f12\u5468\u7684Ib\u671f\u55ae\u5291\u91cf\u7814\u7a76\uff08NCT06679959\uff09\u4e2d\u9032\u884c\u8a55\u4f30\uff0c\u7d50\u679c\u986f\u793a\u5176\u8868\u89c0\u534a\u8870\u671f\uff08observed half-life\uff09\u70ba46\u5929\u81f375\u5929\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A2\u6b64\u524d\u5c1a\u672a\u958b\u5c55\u904e\u4eba\u9ad4\u7814\u7a76\u3002\u5728\u672c\u7814\u7a76\u4e2d\uff0c\u5236\u5291A1\u5728\u80a5\u80d6\u60a3\u8005\u4e2d\u9054\u5230\u4e86\u6cbb\u7642\u6027\u85e5\u7269\u66b4\u9732\u6c34\u5e73\uff08therapeutic drug exposures\uff09\uff0c\u800c\u5236\u5291A2\u672a\u9054\u5230\u3002 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Platform\uff0cULAP\uff09\u6280\u8853\u5728\u958b\u767c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u7684\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7642\u6cd5\u7684\u53ef\u884c\u6027\u3002\u300d \u7531\u6b4c\u79ae\u81ea\u4e3b\u7814\u767c\u7684ASC30\u662f\u9996\u6b3e\u4e5f\u662f\u552f\u4e00\u4e00\u6b3e\u6b63\u5728\u81e8\u5e8a\u7814\u7a76\u4e2d\u7684\u3001\u65e2\u53ef\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u4e5f\u53ef\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u7684\u5c0f\u5206\u5b50GLP-1R\u504f\u5411\u6fc0\u52d5\u5291\uff0c\u65e2\u53ef\u4f5c\u70ba\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\u4e5f\u53ef\u4f5c\u70ba\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u3002 \u95dc\u65bcASC30 ASC30\u662f\u4e00\u6b3e\u6b63\u5728\u81e8\u5e8a\u7814\u7a76\u4e2d\u7684\u5c0f\u5206\u5b50GLP-1R\u504f\u5411\u6fc0\u52d5\u5291\uff0c\u5177\u6709\u7368\u7279\u548c\u5dee\u7570\u5316\u6027\u8cea\uff0c\u4f7f\u5f97\u540c\u4e00\u5c0f\u5206\u5b50\u540c\u6642\u9069\u7528\u65bc\u53e3\u670d\u7247\u5291\u548c\u76ae\u4e0b\u6ce8\u5c04\u7d66\u85e5\u6210\u70ba\u53ef\u80fd\u3002ASC30\u662f\u4e00\u7a2e\u65b0\u5316\u5b78\u5be6\u9ad4\uff08NCE\uff09\uff0c\u64c1\u6709\u7f8e\u570b\u548c\u5168\u7403\u5316\u5408\u7269\u5c08\u5229\u4fdd\u8b77\uff0c\u5c08\u5229\u4fdd\u8b77\u671f\u81f32044\u5e74\uff08\u4e0d\u542b\u6f5b\u5728\u7684\u5c08\u5229\u5ef6\u671f\uff09\u3002 \u95dc\u65bc\u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8 \u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8\u662f\u4e00\u5bb6\u5168\u50f9\u503c\u93c8\u6574\u5408\u578b\u751f\u7269\u6280\u8853\u516c\u53f8\uff0c\u805a\u7126\u6709\u671b\u6210\u70ba\u6cbb\u7642\u4ee3\u8b1d\u75be\u75c5\u540c\u985e\u6700\u4f73\uff08best-in-class\uff09\u548c\u540c\u985e\u9996\u5275\uff08first-in-class\uff09\u85e5\u7269\u7684\u958b\u767c\u548c\u5546\u696d\u5316\u3002\u5229\u7528\u516c\u53f8\u5c08\u6709\u7684\u57fa\u65bc\u7d50\u69cb\u7684AI\u8f14\u52a9\u85e5\u7269\u767c\u73fe\uff08Artificial Intelligence-assisted Structure-Based Drug Discovery\uff0cAISBDD\uff09\u3001\u8d85\u9577\u6548\u85e5\u7269\u958b\u767c\u5e73\u53f0\uff08Ultra-Long-Acting Platform\uff0cULAP\uff09\u6280\u8853\u4ee5\u53ca\u53e3\u670d\u591a\u80bd\u905e\u9001\u589e\u5f37\u6280\u8853\uff08Peptide Oral Transport ENhancement Technology\uff0cPOTENT\uff09\uff0c\u6b4c\u79ae\u5df2\u81ea\u4e3b\u7814\u767c\u591a\u6b3e\u5c0f\u5206\u5b50\u548c\u591a\u80bd\u5019\u9078\u85e5\u7269\uff0c\u5305\u62ec\u5176\u6838\u5fc3\u9805\u76eeASC30\uff0c\u4e00\u6b3e\u5728\u7814\u5c0f\u5206\u5b50GLP-1R\u6fc0\u52d5\u5291\uff0c\u65e2\u53ef\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u4e5f\u53ef\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u4f5c\u70ba\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\u548c\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\uff1bASC36\uff0c\u4e00\u6b3e\u80f0\u6fb1\u7d20\u53d7\u9ad4\u6fc0\u52d5\u5291\u591a\u80bd\uff0cASC35\uff0c\u4e00\u6b3e\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04GLP-1R\/GIPR\u96d9\u9776\u9ede\u6fc0\u52d5\u5291\u591a\u80bd\uff0cASC37\uff0c\u4e00\u6b3eGLP-1R\/GIPR\/GCGR\u4e09\u9776\u9ede\u6fc0\u52d5\u5291\u591a\u80bd\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u3002\u6b4c\u79ae\u5df2\u5728\u9999\u6e2f\u806f\u4ea4\u6240\u4e0a\u5e02\uff081672.HK\uff09\u3002 \u6b32\u77ad\u89e3\u66f4\u591a\u4fe1\u606f\uff0c\u656c\u8acb\u767b\u9304\u7db2\u7ad9\uff1awww.ascletis.com\u3002 \u8a73\u60c5\u5782\u8a62\uff1a Peter VozzoICR Healthcare443-231-0505 (\u7f8e\u570b)Peter.vozzo@icrhealthcare.com \u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8PR\u548cIR\u5718\u968a+86-181-0650-9129 (\u4e2d\u570b)pr@ascletis.comir@ascletis.com\u00a0\" \/>\n<meta property=\"og:url\" content=\"https:\/\/pingtungtimes.com.tw\/?p=416426\" \/>\n<meta property=\"og:site_name\" content=\"\u5c4f\u6771\u6642\u5831\u96fb\u5b50\u5831\" \/>\n<meta property=\"article:publisher\" content=\"https:\/\/www.facebook.com\/pingtungnews\" \/>\n<meta property=\"article:published_time\" content=\"2026-03-10T10:00:00+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/pingtungtimes.com.tw\/wp-content\/uploads\/2023\/02\/logo-150.png\" \/>\n<meta name=\"author\" content=\"\u7f8e\u901a\u793e\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:image\" content=\"https:\/\/pingtungtimes.com.tw\/wp-content\/uploads\/2023\/02\/logo-150.png\" \/>\n<meta name=\"twitter:label1\" content=\"\u4f5c\u8005:\" \/>\n\t<meta name=\"twitter:data1\" content=\"\u7f8e\u901a\u793e\" \/>\n\t<meta name=\"twitter:label2\" content=\"\u9810\u4f30\u95b1\u8b80\u6642\u9593\" \/>\n\t<meta name=\"twitter:data2\" content=\"1 \u5206\u9418\" \/>\n<script type=\"application\/ld+json\" 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kg\\\/m\u00b2\uff09\u4e2d\u7684\u5b89\u5168\u6027\u3001\u8010\u53d7\u6027\u53ca\u7642\u6548\u300265\u4f8b\u53d7\u8a66\u8005\u5747\u5728\u7b2c1\u5929\u3001\u7b2c29\u5929\uff08\u7b2c4\u5468\uff09\u53ca\u7b2c57\u5929\uff08\u7b2c8\u5468\uff09\u63a5\u53d7\u6bcf\u6708\u4e00\u6b21\u7684ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u6216\u5339\u914d\u7684\u5b89\u6170\u5291\u7d66\u85e5\uff08\u51713\u5291\uff09\uff0c\u7121\u9700\u6bcf\u9031\u4e00\u6b21\u7d66\u85e5\u7684\u6e96\u5099\uff08lead-in\uff09\u671f\u3002\u7dad\u6301\u671f\u5f9e\u7b2c8\u5468\u958b\u59cb\u81f3\u7b2c24\u5468\uff0c\u517116\u5468\u3002\u8a72\u7814\u7a76\u5c0dASC30\u7684\u5169\u7a2e\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\uff08A1\u548cA2\uff09\u9032\u884c\u4e86\u8a55\u4f30\uff0c\u7814\u7a76\u76ee\u7684\u70ba\u8a55\u4f30\u6bcf\u6708\u4e00\u6b21\u7d66\u85e5\u7684\u6cbb\u7642\u7642\u6cd5\u548c\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7d66\u85e5\u7684\u7dad\u6301\u7642\u6cd5\u7684\u6f5b\u529b\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u6b64\u524d\u5df2\u5728\u4e00\u9805\u70ba\u671f12\u5468\u7684Ib\u671f\u55ae\u5291\u91cf\u7814\u7a76\uff08NCT06679959\uff09\u4e2d\u9032\u884c\u8a55\u4f30\uff0c\u7d50\u679c\u986f\u793a\u5176\u8868\u89c0\u534a\u8870\u671f\uff08observed half-life\uff09\u70ba46\u5929\u81f375\u5929\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A2\u6b64\u524d\u5c1a\u672a\u958b\u5c55\u904e\u4eba\u9ad4\u7814\u7a76\u3002\u5728\u672c\u7814\u7a76\u4e2d\uff0c\u5236\u5291A1\u5728\u80a5\u80d6\u60a3\u8005\u4e2d\u9054\u5230\u4e86\u6cbb\u7642\u6027\u85e5\u7269\u66b4\u9732\u6c34\u5e73\uff08therapeutic drug exposures\uff09\uff0c\u800c\u5236\u5291A2\u672a\u9054\u5230\u3002 ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u7684\u7d66\u85e5\u65b9\u6848\uff1a\u6240\u6709\u53d7\u8a66\u8005\u63a5\u53d7\u4e09\u6b21\u76ae\u4e0b\u7d66\u85e5\uff0c\u7d66\u85e5\u9593\u9694\u70ba\u56db\u5468\uff0c\u5206\u5225\u5728\u7b2c1\u5929\u3001\u7b2c29\u5929\uff08\u7b2c4\u5468\uff09\u548c\u7b2c57\u5929\uff08\u7b2c8\u5468\uff09\u7d66\u85e5\uff0c\u6bcf\u6b21\u5291\u91cf\u70ba400\u6beb\u514b\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u5728\u7b2c4\u5468\u3001\u7b2c8\u5468\u3001\u7b2c12\u5468\u548c\u7b2c16\u5468\u5206\u5225\u5be6\u73fe\u4e862.7%\u30015.5%\u30016.3%\u548c7.5%\u7684\u7d93\u5b89\u6170\u5291\u6821\u6b63\u5f8c\u7684\u5e73\u5747\u9ad4\u91cd\u4e0b\u964d\u3002\u9019\u4e9b\u6578\u64da\u986f\u793a\uff0cASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u53ef\u6bcf\u6708\u4e00\u6b21\u7d66\u85e5\u7528\u65bc\u80a5\u80d6\u75c7\u6cbb\u7642\uff0c\u4e26\u6709\u671b\u5be6\u73fe\u6bcf\u5169\u500b\u6708\u4e00\u6b21\u7d66\u85e5\uff0c\u4e14\u7121\u9700\u6bcf\u9031\u4e00\u6b21\u7d66\u85e5\u7684\u6e96\u5099\u671f\u3002 \u8a72II\u671f\u7814\u7a76\u540c\u6642\u8a55\u4f30\u4e86ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u4f5c\u70ba\u7dad\u6301\u7642\u6cd5\u7684\u6f5b\u529b\u3002\u5728\u7b2c8\u5468\u5b8c\u6210\u672b\u6b21\u7d66\u85e5\u5f8c\uff0c\u5c0d\u5728\u60a3\u8005\u4e2d\u7684\u7642\u6548\u6301\u7e8c\u6642\u9593\u9032\u884c\u4e86\u70ba\u671f16\u5468\u7684\u8a55\u4f30\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u5728\u672b\u6b21\u7d66\u85e5\u5f8c\u768416\u5468\u7dad\u6301\u671f\u5167\u5747\u9054\u5230\u4e86\u6cbb\u7642\u6027\u85e5\u7269\u66b4\u9732\u6c34\u5e73\u3002\u7d93\u5b89\u6170\u5291\u6821\u6b63\u5f8c\u7684\u5e73\u5747\u9ad4\u91cd\u4e0b\u964d\u5728\u7b2c8\u5468\u70ba5.5%\uff0c\u7b2c20\u5468\uff08\u672b\u6b21\u7d66\u85e5\u5f8c3\u500b\u6708\uff09\u70ba6.4%\uff0c\u7b2c24\u5468\uff08\u672b\u6b21\u7d66\u85e5\u5f8c4\u500b\u6708\uff09\u70ba5.8%\u3002\u9019\u4e9b\u7d50\u679c\u986f\u793aASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u6709\u671b\u6210\u70ba\u6bcf\u5b63\u5ea6\u7d66\u85e5\u4e00\u6b21\u7684\u6709\u6548\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\u3002 ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u548cA2\u5b89\u5168\u6027\u548c\u8010\u53d7\u6027\u826f\u597d\uff0c\u5176\u5b89\u5168\u6027\u548c\u8010\u53d7\u6027\u7279\u5fb5\u548cGLP\u20111\u985e\u85e5\u7269\u4e00\u81f4\u3002\u7d93ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u548cA2\u6216\u5b89\u6170\u5291\u6cbb\u7642\u7684\u53d7\u8a66\u8005\u5747\u7121\u56e0\u4e0d\u826f\u4e8b\u4ef6\uff08AE\uff09\u800c\u505c\u85e5\u7684\u60c5\u6cc1\u3002\u6240\u6709\u4e0d\u826f\u4e8b\u4ef6\uff08\u5305\u62ec\u6ce8\u5c04\u90e8\u4f4d\u4e0d\u826f\u4e8b\u4ef6\uff09\u7684\u56b4\u91cd\u7a0b\u5ea6\u5747\u70ba\u8f15\u5ea6\u81f3\u4e2d\u5ea6\u3002\u6240\u6709\u80c3\u8178\u9053\uff08GI\uff09\u4e0d\u826f\u4e8b\u4ef6\u5747\u70ba\u8f15\u5ea6\uff081\u7d1a\uff09\uff0c\u7121\u4e2d\u5ea6\uff082\u7d1a\uff09\u53ca\u4ee5\u4e0a\u80c3\u8178\u9053\u4e0d\u826f\u4e8b\u4ef6\u3002\u672a\u89c0\u5bdf\u5230\u809d\u81df\u5b89\u5168\u6027\u4fe1\u865f\u3002\u6b64\u5916\uff0c\u5be6\u9a57\u5ba4\u6aa2\u67e5\u3001\u751f\u547d\u9ad4\u5f81\u3001\u5fc3\u96fb\u5716\uff08\u5305\u62ecQTc\u9593\u671f\uff09\u548c\u9ad4\u683c\u6aa2\u67e5\u5747\u672a\u898b\u7570\u5e38\u7d50\u679c\u3002 \u300c\u5728\u63a5\u53d7ASC30\u9577\u6548\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u6cbb\u7642\u7684\u80a5\u80d6\u60a3\u8005\u4e2d\u89c0\u5bdf\u5230\u5177\u6709\u7d71\u8a08\u5b78\u986f\u8457\u6027\u548c\u81e8\u5e8a\u610f\u7fa9\u7684\u9ad4\u91cd\u4e0b\u964d\uff0c\u6211\u5011\u6df1\u611f\u632f\u596e\u3002ASC30\u65e2\u53ef\u4f5c\u70ba\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u7d66\u85e5\u6216\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u7d66\u85e5\u7684\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\uff0c\u4e5f\u53ef\u4f5c\u70ba\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u7d66\u85e5\u7684\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u662f\u9996\u6b3e\u4e5f\u662f\u552f\u4e00\u4e00\u6b3e\u64c1\u6709\u4e0a\u8ff0\u7d66\u85e5\u983b\u7387\u548c\u7d66\u85e5\u9014\u5f91\u4e26\u5df2\u5728\u5169\u9805II\u671f\u7814\u7a76\u4e2d\u8b49\u660e\u53ef\u5be6\u73fe\u6709\u6548\u6e1b\u91cd\u7684\u8178\u4fc3\u80f0\u7d20\uff08incretin\uff09\u3002\u300d\u6b4c\u79ae\u5275\u59cb\u4eba\u3001\u8463\u4e8b\u6703\u4e3b\u5e2d\u517c\u9996\u5e2d\u57f7\u884c\u5b98\u5433\u52c1\u6893\u535a\u58eb\u8868\u793a\uff0c\u300cASC30\u9577\u6548\u5236\u5291\u517c\u5177\u5177\u6709\u7af6\u722d\u529b\u7684\u7642\u6548\u8207\u826f\u597d\u7684\u5b89\u5168\u6027\u3001\u8010\u53d7\u6027\u7279\u5fb5\uff0c\u9019\u9032\u4e00\u6b65\u589e\u5f37\u4e86\u6211\u5011\u64f4\u5927ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u81e8\u5e8a\u958b\u767c\u9805\u76ee\u7684\u4fe1\u5fc3\uff0c\u5305\u62ec\u6bcf\u6708\u4e00\u6b21\u7684\u6cbb\u7642\u7642\u6cd5\uff0c\u4ee5\u53ca\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7684\u7dad\u6301\u7642\u6cd5\u3002\u6b64\u5916\uff0c\u5f9e\u9019\u9805\u70ba\u671f24\u5468\u3001\u4f7f\u7528\u6b4c\u79ae\u5c08\u6709\u7684\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u7684\u7814\u7a76\u4e2d\u7372\u5f97\u7684\u6578\u64da\uff0c\u9a57\u8b49\u4e86\u6b4c\u79ae\u8d85\u9577\u6548\u85e5\u7269\u958b\u767c\u5e73\u53f0\uff08Ultra-Long-Acting Platform\uff0cULAP\uff09\u6280\u8853\u5728\u958b\u767c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u7684\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7642\u6cd5\u7684\u53ef\u884c\u6027\u3002\u300d \u7531\u6b4c\u79ae\u81ea\u4e3b\u7814\u767c\u7684ASC30\u662f\u9996\u6b3e\u4e5f\u662f\u552f\u4e00\u4e00\u6b3e\u6b63\u5728\u81e8\u5e8a\u7814\u7a76\u4e2d\u7684\u3001\u65e2\u53ef\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u4e5f\u53ef\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u7684\u5c0f\u5206\u5b50GLP-1R\u504f\u5411\u6fc0\u52d5\u5291\uff0c\u65e2\u53ef\u4f5c\u70ba\u6e1b\u91cd\u6cbb\u7642\u7642\u6cd5\u4e5f\u53ef\u4f5c\u70ba\u6e1b\u91cd\u7dad\u6301\u7642\u6cd5\uff0c\u7528\u65bc\u9577\u671f\u9ad4\u91cd\u7ba1\u7406\u3002 \u95dc\u65bcASC30 ASC30\u662f\u4e00\u6b3e\u6b63\u5728\u81e8\u5e8a\u7814\u7a76\u4e2d\u7684\u5c0f\u5206\u5b50GLP-1R\u504f\u5411\u6fc0\u52d5\u5291\uff0c\u5177\u6709\u7368\u7279\u548c\u5dee\u7570\u5316\u6027\u8cea\uff0c\u4f7f\u5f97\u540c\u4e00\u5c0f\u5206\u5b50\u540c\u6642\u9069\u7528\u65bc\u53e3\u670d\u7247\u5291\u548c\u76ae\u4e0b\u6ce8\u5c04\u7d66\u85e5\u6210\u70ba\u53ef\u80fd\u3002ASC30\u662f\u4e00\u7a2e\u65b0\u5316\u5b78\u5be6\u9ad4\uff08NCE\uff09\uff0c\u64c1\u6709\u7f8e\u570b\u548c\u5168\u7403\u5316\u5408\u7269\u5c08\u5229\u4fdd\u8b77\uff0c\u5c08\u5229\u4fdd\u8b77\u671f\u81f32044\u5e74\uff08\u4e0d\u542b\u6f5b\u5728\u7684\u5c08\u5229\u5ef6\u671f\uff09\u3002 \u95dc\u65bc\u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8 \u6b4c\u79ae\u88fd\u85e5\u6709\u9650\u516c\u53f8\u662f\u4e00\u5bb6\u5168\u50f9\u503c\u93c8\u6574\u5408\u578b\u751f\u7269\u6280\u8853\u516c\u53f8\uff0c\u805a\u7126\u6709\u671b\u6210\u70ba\u6cbb\u7642\u4ee3\u8b1d\u75be\u75c5\u540c\u985e\u6700\u4f73\uff08best-in-class\uff09\u548c\u540c\u985e\u9996\u5275\uff08first-in-class\uff09\u85e5\u7269\u7684\u958b\u767c\u548c\u5546\u696d\u5316\u3002\u5229\u7528\u516c\u53f8\u5c08\u6709\u7684\u57fa\u65bc\u7d50\u69cb\u7684AI\u8f14\u52a9\u85e5\u7269\u767c\u73fe\uff08Artificial Intelligence-assisted Structure-Based Drug Discovery\uff0cAISBDD\uff09\u3001\u8d85\u9577\u6548\u85e5\u7269\u958b\u767c\u5e73\u53f0\uff08Ultra-Long-Acting Platform\uff0cULAP\uff09\u6280\u8853\u4ee5\u53ca\u53e3\u670d\u591a\u80bd\u905e\u9001\u589e\u5f37\u6280\u8853\uff08Peptide Oral Transport ENhancement 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kg\/m\u00b2\uff09\u4e2d\u7684\u5b89\u5168\u6027\u3001\u8010\u53d7\u6027\u53ca\u7642\u6548\u300265\u4f8b\u53d7\u8a66\u8005\u5747\u5728\u7b2c1\u5929\u3001\u7b2c29\u5929\uff08\u7b2c4\u5468\uff09\u53ca\u7b2c57\u5929\uff08\u7b2c8\u5468\uff09\u63a5\u53d7\u6bcf\u6708\u4e00\u6b21\u7684ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\u6216\u5339\u914d\u7684\u5b89\u6170\u5291\u7d66\u85e5\uff08\u51713\u5291\uff09\uff0c\u7121\u9700\u6bcf\u9031\u4e00\u6b21\u7d66\u85e5\u7684\u6e96\u5099\uff08lead-in\uff09\u671f\u3002\u7dad\u6301\u671f\u5f9e\u7b2c8\u5468\u958b\u59cb\u81f3\u7b2c24\u5468\uff0c\u517116\u5468\u3002\u8a72\u7814\u7a76\u5c0dASC30\u7684\u5169\u7a2e\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291\uff08A1\u548cA2\uff09\u9032\u884c\u4e86\u8a55\u4f30\uff0c\u7814\u7a76\u76ee\u7684\u70ba\u8a55\u4f30\u6bcf\u6708\u4e00\u6b21\u7d66\u85e5\u7684\u6cbb\u7642\u7642\u6cd5\u548c\u6bcf\u5b63\u5ea6\u4e00\u6b21\u7d66\u85e5\u7684\u7dad\u6301\u7642\u6cd5\u7684\u6f5b\u529b\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A1\u6b64\u524d\u5df2\u5728\u4e00\u9805\u70ba\u671f12\u5468\u7684Ib\u671f\u55ae\u5291\u91cf\u7814\u7a76\uff08NCT06679959\uff09\u4e2d\u9032\u884c\u8a55\u4f30\uff0c\u7d50\u679c\u986f\u793a\u5176\u8868\u89c0\u534a\u8870\u671f\uff08observed half-life\uff09\u70ba46\u5929\u81f375\u5929\u3002ASC30\u76ae\u4e0b\u5132\u5eab\u578b\u5236\u5291A2\u6b64\u524d\u5c1a\u672a\u958b\u5c55\u904e\u4eba\u9ad4\u7814\u7a76\u3002\u5728\u672c\u7814\u7a76\u4e2d\uff0c\u5236\u5291A1\u5728\u80a5\u80d6\u60a3\u8005\u4e2d\u9054\u5230\u4e86\u6cbb\u7642\u6027\u85e5\u7269\u66b4\u9732\u6c34\u5e73\uff08therapeutic drug exposures\uff09\uff0c\u800c\u5236\u5291A2\u672a\u9054\u5230\u3002 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